Setiptiline maleate
CAS No. 85650-57-3
Setiptiline maleate ( MO-8282 )
产品货号. M16210 CAS No. 85650-57-3
A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥640 | 有现货 |
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50MG | ¥2908 | 有现货 |
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100MG | ¥4196 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Setiptiline maleate
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist.
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产品描述A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, as well as an H1 receptor inverse agonist/antihistamine.Depression Approved
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同义词MO-8282
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT Receptor
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研究领域Neurological Disease
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适应症Depression
化学信息
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CAS Number85650-57-3
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分子量377.43
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分子式C23H23NO4
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纯度>98% (HPLC)
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溶解度10 mM in DMSO
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SMILESCN1CCC2=C(C1)C3=CC=CC=C3CC4=CC=CC=C24.C(=CC(=O)O)C(=O)O
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化学全称1H-Dibenzo[3,4:6,7]cyclohepta[1,2-c]pyridine, 2,3,4,9-tetrahydro-2-methyl-, (2Z)-2-butenedioate (1:1)
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Niho T, et al. Nihon Yakurigaku Zasshi. 1986 Oct;88(4):309-20.
2. Mizota M, et al. Nihon Yakurigaku Zasshi. 1986 Dec;88(6):457-66.
3. Przegaliński E, et al. Pol J Pharmacol Pharm. 1986 Jul-Aug;38(4):377-84.
2. Mizota M, et al. Nihon Yakurigaku Zasshi. 1986 Dec;88(6):457-66.
3. Przegaliński E, et al. Pol J Pharmacol Pharm. 1986 Jul-Aug;38(4):377-84.
产品手册
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